Synthesis of irreversibly binding bicalutamide analogs for imaging studies

Vipin A Nair; Suni M Mustafa; Michael L Mohler; Jun Yang; Leonid I Kirkovsky; James T Dalton; Duane D Miller

doi:10.1016/j.tetlet.2005.04.143

Synthesis of irreversibly binding bicalutamide analogs for imaging studies

Tetrahedron Lett. 2005 Jul 11;46(28):4821-4823. doi: 10.1016/j.tetlet.2005.04.143.

Authors

Vipin A Nair¹, Suni M Mustafa, Michael L Mohler, Jun Yang, Leonid I Kirkovsky, James T Dalton, Duane D Miller

Affiliation

¹ Department of Pharmaceutical Sciences, University of Tennessee, The Health Science Center, 847 Monroe Avenue, RM 227 C, Memphis, TN 38163, USA.

Abstract

A new synthetic methodology for preparing radioactive androgen receptor binding compounds in order to determine receptor-ligands interactions has been developed.

Abstract

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