Inverse agonism at G protein-coupled receptors: (patho)physiological relevance and implications for drug discovery

Br J Pharmacol. 2000 May;130(1):1-12. doi: 10.1038/sj.bjp.0703311.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Calcium Channel Agonists / pharmacology*
  • Calcium Channels / drug effects*
  • Calcium Channels / physiology
  • Drug Design
  • GTP-Binding Proteins / agonists*
  • GTP-Binding Proteins / physiology
  • Humans
  • Receptors, Cell Surface / agonists*
  • Receptors, Cell Surface / physiology
  • Receptors, Drug / agonists*
  • Receptors, Drug / physiology

Substances

  • Calcium Channel Agonists
  • Calcium Channels
  • Receptors, Cell Surface
  • Receptors, Drug
  • GTP-Binding Proteins