Associate editor: H. BönischCytochrome P450 enzymes in drug metabolism: Regulation of gene expression, enzyme activities, and impact of genetic variation
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Keywords
Biotransformation
Cytochrome P450 monooxygenase
NADPH:cytochrome P450 reductase
Pharmacogenetics
Polymorphism
Xenobiotic
Abbreviations
ADME
absorption, distribution, metabolism, excretion
ADR
adverse drug reaction
AhR
aromatic hydrocarbon receptor
CNV
copy number variant
CYP
cytochrome P450
DDI
drug-drug interaction
EM
extensive metabolizer
ERα
estrogen receptor alpha
FXR
farnesoid X receptor
GR
glucocorticoid receptor
GWAS
genome-wide association study
IM
intermediate metabolizer
LD
linkage disequilibrium
LXR
liver X receptor
MAF
minor allele frequency
NAFLD
non-alcoholic fatty liver disease
NASH
non-alcoholic steatohepatitis
NNRTI
non-nucleoside reverse transcriptase inhibitor
PBREM
phenobarbital-responsive enhancer module
PCR
polymerase chain reaction
PM
poor metabolizer
POR
NADPH:cytochrome P450 oxidoreductase
PPAR
peroxisome proliferator-activated receptor
SERM
selective estrogen receptor modulator
SLCO1B1
organic anion transporting polypeptide 1B1
UM
ultrarapid metabolizer
VDR
vitamin D receptor
XREM
xenobiotics-responsive enhancer module
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