Pharmacological characterization of [D-Ala2,Leu5,Ser6]enkephalin (DALES): antinociceptive actions at the δnon-complexed-opioid receptor
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Cited by (13)
Quantitative autoradiographic mapping of opioid receptors in the brain of δ-opioid receptor gene knockout mice
2002, Brain ResearchCitation Excerpt :It is worthy of note that those regions in heterozygous mice that show rather less than 50% loss of δ-receptors (e.g., habenula, lateral septum and superior colliculus) are also regions which have a high level of μ-receptors and thus a proportion of the binding measured is probably due to μ-cross labeling. There is substantial pharmacological and molecular evidence to suggest heterogeneity of δ-receptors [10,14,18,25,26,28,44]. Only a single gene, Oprd1, has been identified encoding the δ-receptor although the cloned receptor has been reported to exhibit higher affinity for putative δ2-receptor selective ligands than for δ1-selective compounds [31].
Novel met-enkephalin analogue: A potent systemic mu agonist antinociceptive agent
1995, Pharmacological ResearchIdentification of a human delta opioid receptor: Cloning and expression
1994, Life SciencesPseudoirreversible binding characteristics of [D-Ala<sup>2</sup>, Glu<sup>4</sup>]deltorphin and its Cys<sup>4</sup> substituted derivative to δ-opioid receptors
1993, European Journal of Pharmacology: Molecular Pharmacology
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