TABLE 3

Cmax (±S.E.M.) and AUC values for OEA and KDS-5104 (analog 3) after oral administration (100 mg kg–1)



Plasma

Liver

Cmax
AUC
Cmax
AUC
μg ml–1 μg min ml–1 μg g–1 wet tissue μg min g–1
OEA 0.07 ± 0.01 18.42 0.16 ± 0.03 58.51
KDS-5104
0.58 ± 0.06
198.13
2.92 ± 0.79
674.12