TABLE 1

Specificity of SD-282 for p38 MAPK isoforms


Kinase Target

IC50
SD-282
Control
μmol / l
p38α 0.00161 0.022*
p38β 0.023 0.028*
p38γ >10 μM 0.57**
p38δ
>10 μM
0.36**
  • * SB 202190

  • ** Staurosporine