TABLE 1
Specificity of SD-282 for p38 MAPK isoforms
Kinase Target
IC
50
SD-282
Control
μ
mol / l
p38α
0.00161
0.022
*
p38β
0.023
0.028
*
p38γ
>10 μM
0.57
**
p38δ
>10 μM
0.36
**
↵
*
SB 202190
↵
**
Staurosporine