Enzyme | IC50 | Enzyme | IC50 | Enzyme | IC50 |
---|---|---|---|---|---|
μM | μM | μM | |||
IKKα | >100 | PKCα | >100 | ERK2 | >100 |
IKKϵ | >100 | PKCδ | 50 | p38a | >100 |
PKA | >100 | PKCθ | 50 | MKK6 | >83 |
CaM KII | >100 | CSK | >50 | MEK1 | >83 |
CDK2/cyclin E | >100 | Src | >50 | cRaf-1 | >83 |
CKII | >100 | Lyn | >50 | cABL1 | >50 |
LCK | >100 | MK2 | >50 | p70 S6K | >100 |
CHK1 | >100 | KDR | >50 | ROKA | >100 |
MAPKAPPK2 | >100 | JNK1 | 84 | SGK1 | >100 |
PLK | >100 | PRPK | >100 | PRAK | >100 |