TABLE 2
K
i
for inhibitors at various kinases
Inhibitor
PKA
PKG
PKC
ROCK
μ
M
Y-27632
25
26
0.1
HA-1077
1.6
1.6
0.33
Chelerytherine
0.66
H7
3
5.8
6
0.45
H89
0.05
0.5
0.27