TABLE 2

Ki for inhibitors at various kinases


Inhibitor

PKA

PKG

PKC

ROCK
μM
Y-27632 25 26 0.1
HA-1077 1.6 1.6 0.33
Chelerytherine 0.66
H7 3 5.8 6 0.45
H89
0.05
0.5

0.27