Cockroach GluCl-Da | Cockroach GluCl-Nb | Cockroach GABA-Rs | Rat DRG GABAA-Rs | |
---|---|---|---|---|
Fipronil sulfone | ||||
IC50 (nM) | ||||
Uc | 350 | 31.2, 12.3, 8.8d | 53.7, 26.6, 15.4d | 46.6, 20d |
B/Ue | 25 | 8.5 | 20 | 70.2 |
EBOBf | 9 (insect mean) | 175 (vertebrate mean) | ||
Fipronil | ||||
IC50 (nM) | ||||
U | 750 | 27, 17.3, 11.9g | 35 | 1610h |
B/U | 801i | 10i | 27.6g | Not applicable |
EBOBf |
|
| 7.0 (insect mean) | 1103 (vertebrate mean) |