TABLE 2

GI50 on various cancer cells


Cell Lines

Tumor Types

GI50
μM
NCI H322M NSCLC 0.35
NCI H460 NSCLC 1.62
NCI H522 NSCLC 1.95
HCT-116 Colon cancer 0.41
KM12 Colon cancer 0.13
SF-295 CNS cancer 0.04
SF-268 CNS cancer 2.29
M14 Melanoma 1.20
IGROV1 Ovarian cancer 0.44
OVCAR-3 Ovarian cancer 0.07
OVCAR-5 Ovarian cancer 1.95
NCI/ADR-RES
Breast cancer
0.41