Reference/Source | (—)-Cocaine vs. [3H]DA (IC50) | (—)-Cocaine vs. [3H]PEA (IC50) | DAT Source | |
---|---|---|---|---|
nM | ||||
Current results | 167 | 19.8 | Human DAT in HEK cells | |
Yatin et al. (2002) | 221 | Human DAT in HEK cells | ||
Eshleman et al. (1999) | 278 | Human DAT in HEK cells | ||
Calligaro and Eldefrawi (1987) | 770 | Rat striatal synaptosomes | ||
Debler et al. (1988) | 200 | Mouse striatal synaptosomes | ||
Hyttel (1978) | 310 | Rat striatal synaptosomes | ||
Matecka et al. (1996) | 478 |
| Rat striatal synaptosomes |