TABLE 3

Ancillary receptor binding affinities determined for WAY-163909

Data are average values obtained in two independent experiments using human receptor subtypes (except *rat cortical membranes) expressed in stable CHO cell lines.


Receptor

Ki
nM
5-HT1A >1000
5-HT7 343
D2 >1000
D3 >1000
D4 245
5-HT-T* >1000
α-1*
665