Drug | IC50a | Maximum Inhibition | ||
---|---|---|---|---|
Con | % Inhibition | |||
μM (95 % CI) | μM | Mean ± S.E.M. | ||
100 μM (−)-Nicotine-[3H]DA | ||||
Mec | 0.20 (0.07, 0.57) | 100 | 86 ± 10 | |
MG 624 | 0.54 (0.18, 1.59) | 100 | 60 ± 11 | |
Hex | 3.16 (0.53, 18.9) | 1000 | 87 ± 6 | |
d-TC | 6.31 (1.87, 21.3) | 1000 | 79 ± 8 | |
DHβE | 61 (21, 183) | 1000 | 67 ± 10 | |
MLA | N.D. | 0.010 | −4 ± 6 | |
α-CtxImI | N.D. | 1.0 | −4 ± 11 | |
α-BTX | N.D. | 0.4 | −1.0 ± 0.9 | |
α-CtxMII | N.D. | 0.1 | 12 ± 14 | |
100 μM (−)-Nicotine-[3H]NE | ||||
MG 624 | 0.34 (0.17, 0.69) | 10 | 111 ± 5 | |
10 μM (±)-UB-165-[3H]NE | ||||
MG 624 | 0.42 (0.22, 0.80) | 10 | 100 ± 5 |
N.D., not able to determine; CI, confidence interval; Con., concentration tested.
↵ a Calculated from pIC50:IC50 = 10−pIC50.