TABLE 1

Affinity (Ki, nM) of ligands for 5-HT2R subtypes


Ligand

Receptor Subtype

Reference
5-HT2AR
5-HT2BR
5-HT2CR
BW 723C86 >3891 12 125 Baxter et al. (1995)
DOI 50a 39a 15a Kennett (1993)
MK 212 15,848 1258 630 Kennett (1993)
SB 204741 5011 15 >1000 Baxter et al. (1995)
SR 46349B 5.8b >100 120b Rinaldi-Carmona et al. (1992)
SDZ SER-082
630c
58
15c
Nozulak et al. (1995)
  • a EC50 (nM).

  • b IC50 (nM).

  • c KD (nM).