IC50 (nM) | |||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Human PARP Inhibition | Mouse PARP Inhibition | [3H]Spiperone Binding | DAT Binding | TBARS | MAO | NOS | |||||||
FR261529 | 33 ± 0.9 | 35 ± 1.1 | >10,000 | >10,000 | >10,000 | >10,000 | >10,000 | ||||||
3-AB | 11,200 ± 810 | 11,800 ± 690 | >10,000 | >10,000 | >10,000 | >10,000 | >10,000 | ||||||
Reference | Apomorphine | Nomifensine | Vitamin E | Pargyline | 7-NID | ||||||||
|
|
| 223 ± 8.7 | 201 ± 6.8 | 228 ± 8.1 | 146 ± 5.1 | 319 ± 5.7 |