Inhibitor | Ki Values | ||
---|---|---|---|
l-[3H]Proline Uptake | [3H]Glycine Uptake | ||
mM | |||
l-Proline | 1.6 ± 0.04 | 2.2 ± 0.2 | |
d-Proline | 1.2 ± 0.3 | 1.9 ± 0.1 | |
cis-4-Hydroxy-l-proline | 30 ± 4 | ∼ 45 ± 13 | |
cis-4-Hydroxy-d-proline | 3.5 ± 0.1 | 3.2 ± 0.2 | |
trans-4-Hydroxy-l-proline | 9.0 ± 0.9 | 5.3 ± 0.6 | |
l-Azetidine-2-carboxylic acid | 1.8 ± 0.1 | 1.9 ± 0.4 | |
3-Amino-1-propanesulfonic acid | 7.1 ± 0.6 | 10.5 ± 0.5 | |
Glycine | 5.1 ± 0.9 | 9.2 ± 1.0 | |
N-Methyl-l-alanine | 2.2 ± 0.1 | 2.0 ± 0.1 |