Ki | |||||
---|---|---|---|---|---|
hDOR | HMOR | hKOR | |||
nM | |||||
SB-235863 | 4.81 ± 00.39 | 906 ± 141 | 249 ± 73 | ||
TAN-67 | 0.85 ± 0.01 | 61.1 ± 16.7 | 201 ± 46 | ||
DPDPE | 4.59 ± 0.59 | 248 ± 55 | >10,000 | ||
Naltrindole | 0.24 ± 0.02 | 7.23 ± 1.71 | 4.36 ± 0.49 | ||
Morphine | 299 ± 8 | 2.98 ± 0.28 | 63.8 ± 10.5 | ||
DAMGO | 1587 ± 165 | 1.83 ± 0.41 | 553.2 ± 67.1 | ||
β-FNA | 10.9 ± 1.7 | 0.44 ± 0.05 | 0.73 ± 0.14 | ||
BRL-52656 | >5000 | 238 ± 5 | 0.23 ± 0.05 | ||
U69593 | >2500 | 331 ± 0.62 | 1.37 ± 0.20 | ||
nor-BNI | 2.86 ± 0.9 | 23.13 ± 0.62 | 0.41 ± 0.11 |