Table 1

Alanine-scanned C-terminal orexin-A-peptides

Position of ReplacementSequence
Orexin-A14–33 CRLYELLHGAGNHAAGILTL-amide
Orexin-A14–33C14AARLYELLHGAGNHAAGILTL-amide
Orexin-A14–33R15ACALYELLHGAGNHAAGILTL-amide
Orexin-A14–33L16ACRAYELLHGAGNHAAGILTL-amide
Orexin-A14–33Y17ACRLAELLHGAGNHAAGILTL-amide
Orexin-A14–33F18ACRLYALLHGAGNHAAGILTL-amide
Orexin-A14–33L19ACRLYEALHGAGNHAAGILTL-amide
Orexin-A14–33L20ACRLYELAHGAGNHAAGILTL-amide
Orexin-A14–33H21ACRLYELLAGAGNHAAGILTL-amide
Orexin-A14–33G22ACRLYELLHAAGNHAAGILTL-amide
Orexin-A14–33G24ACRLYELLHGAANHAAGILTL-amide
Orexin-A14–33N25ACRLYELLHGAGAHAAGILTL-amide
Orexin-A14–33H26ACRLYELLHGAGNAAAGILTL-amide

The replaced amino acid is shown in bold.