Table 5

Stability of DVL2DAL5LanEnk, DPDPE, and Leu-Enkephalin against degradation by rat brain homogenate

Compoundkobst1/2Regression Coefficient (R2)
DVL 2DAL 5LanEnkNo degradation
DPDPENo degradation
Leu-enkephalin1.03 × 10−1 (1/min)6.7 (min)0.998 (1/min)