h5-HT1A | h5-HT1B | h5-HT1D | h5-HT2A | h5-HT2B | h5-HT2C | H1 | |
---|---|---|---|---|---|---|---|
Apomorphine | 6.93 ± 0.12 | 5.53 ± 0.06 | 5.91 ± 0.15 | 6.92 ± 0.06 | 6.88 ± 0.15 | 6.99 ± 0.07 | <5 |
Bromocriptine | 7.89 ± 0.04 | 6.45 ± 0.12 | 7.97 ± 0.03 | 6.97 ± 0.15 | 7.25 ± 0.07 | 6.13 ± 0.04 | <5 |
Cabergoline | 7.70 ± 0.17 | 6.32 ± 0.09 | 8.06 ± 0.08 | 8.21 ± 0.08 | 8.93 ± 0.016-a | 6.16 ± 0.02 | 5.86 ± 0.14 |
Lisuride | 9.83 ± 0.05 | 7.73 ± 0.11 | 9.01 ± 0.05 | 8.56 ± 0.03 | 8.88 ± 0.05 | 8.18 ± 0.02 | 7.46 ± 0.04 |
Pergolide | 8.72 ± 0.13 | 6.55 ± 0.10 | 7.88 ± 0.11 | 8.08 ± 0.06 | 8.15 ± 0.04 | 6.53 ± 0.06 | 5.77 ± 0.136-a |
Piribedil | 6.35 ± 0.01 | <5 | <5 | <5 | 5.92 ± 0.06 | <5 | <5 |
Pramipexole | 6.16 ± 0.02 | 5.08 ± 0.05 | 5.78 ± 0.10 | <5 | <5 | <5 | <5 |
Quinelorane | <5 | <5 | <5 | <5 | <5 | 5.58 ± 0.12 | 5.98 ± 0.05 |
Quinpirole | 5.77 ± 0.10 | <5 | <5 | <5 | <5 | <5 | 5.98 ± 0.01 |
Ropinirole | 6.54 ± 0.07 | <5 | 5.86 ± 0.07 | <5 | 5.42 ± 0.15 | <5 | 5.53 ± 0.03 |
Roxindole | 9.94 ± 0.24 | 5.84 ± 0.13 | 7.20 ± 0.11 | 8.18 ± 0.01 | 7.51 ± 0.05 | 6.51 ± 0.05 | 6.89 ± 0.076-a |
Talipexole | 5.77 ± 0.04 | <5 | <5 | <5 | <5 | <5 | <5 |
Terguride | 8.46 ± 0.11 | 6.59 ± 0.09 | 7.79 ± 0.15 | 8.32 ± 0.12 | 8.15 ± 0.10 | 7.32 ± 0.07 | 6.47 ± 0.156-a |
TL99 | 5.42 ± 0.06 | <5 | 5.71 ± 0.03 | 5.63 ± 0.07 | 5.69 ± 0.266-a | 5.64 ± 0.21 | 6.11 ± 0.206-a |
Data are pKi values (minus log Kivalues) and, unless, indicated, are expressed as means ± S.E.M. values of at least three independent determinations carried out in triplicate.
↵6-a Mean ± range, n = 2.