Table 2

Relaxation of K+ (20 mM)-stimulated guinea pig bladder smooth muscle strips by adenosine receptor agonists

Compound−log IC50Efficacyn
%
2-Chloroadenosine5.9  ± 0.3279  ± 5.44
NECA6.41  ± 0.0575  ± 64
CGS-216806.38  ± 0.2280  ± 7.34
CPCA6.91  ± 0.1595  ± 3.94
2-Phenylamino adenosine5.53  ± 0.2159  ± 7.54
2Cl-IBMECA>4.5Inactive4
CCPA>4.5Inactive4