Transporter | Potential-Driven | Proton-Driven | Transports TEA | Cimetidine Inhibitable | References |
---|---|---|---|---|---|
OCT1 | Yes | No | Yes | Yes | Gorboulev et al., 1997; Urakami et al., 1998 |
OCT2 | Yes | No | Yes | Yes | Gorboulev et al., 1997; Okuda et al., 1999; Sweet and Pritchard, 1999 |
OCT3 | Yes | No | Yes | Yes | Kekuda et al., 1998; Wu et al., 1998a |
OCTN1 | No | Yes | Yes | Yes | Tamai et al., 1997;Yabuuchi et al., 1999 |
OCTN2 | —1-a | — | Yes | Yes | Wu et al., 1998b, 1999 |
Verapamil transporter | No | Yes | No | No | This study |
↵1-a —, data unavailable.