Table 1

Comparison between cloned organic cation transporters and the RPE cell verapamil transporter

TransporterPotential-DrivenProton-DrivenTransports TEACimetidine InhibitableReferences
OCT1YesNoYesYes Gorboulev et al., 1997; Urakami et al., 1998
OCT2YesNoYesYes Gorboulev et al., 1997; Okuda et al., 1999; Sweet and Pritchard, 1999
OCT3YesNoYesYes Kekuda et al., 1998; Wu et al., 1998a
OCTN1NoYesYesYes Tamai et al., 1997;Yabuuchi et al., 1999
OCTN21-a YesYes Wu et al., 1998b, 1999
Verapamil transporterNoYesNoNoThis study
  • 1-a  —, data unavailable.