Compound | Dose Range | Maximum Substitution | No. Substituted/ No. Tested | Maximum Antagonism | No. Antagonized/ No. Tested |
---|---|---|---|---|---|
mg/kg | % | % | |||
Quinine | 30.0–100.0 | 1.1 at 56.0 | 0 /4 | ||
Linopiridine | 0.1–5.6 | 24.6 at 5.6 | 1 /4 | ||
(±)-BAY K 8644 | 0.3–1.0 | 0.9 at 1.0 | 0 /4 | ||
Pinacidil | 0.03–1.0 | 25.0 at 0.3 | 1 /4 | ||
Cromakalim | 0.01–1.0 | 40.0 at 0.01 | 2 /5 |