Class | Drug | ID50 | 95% CL | MOI | Dose |
---|---|---|---|---|---|
% | mg/kg s.c. | ||||
α2-AR antagonist | Atipamezole | 0.09 | 0.03–0.20 | 91 | 0.63 |
RX821,002 | 0.13 | 0.05–0.30 | 92 | 0.63 | |
Idazoxan | 0.21 | 0.04–1.10 | 99 | 10.0 | |
D1antagonist | NNC756 | 0.02 | 0.01–0.03 | 100 | 0.16 |
SCH23390 | 0.03 | 0.002–0.40 | 98 | 0.16 | |
SCH39166 | 0.17 | 0.06–0.40 | 88 | 0.63 |
95% CL, 95% confidence limits; MOI, maximal observed inhibition.