Ligand | DCUKA IC50 | Ligand | DCUKA IC50 |
---|---|---|---|
μM | μM | ||
[3H]CGP39653 | >200 (19.1 ± 2.1) | [3H]flunitrazepam | >200 (43.6 ± 2.0) |
[3H]Ifenprodil | >200 (9.9 ± 3.7) | [3H]flumazenil | >200 (16.8 ± 4.7) |
[3H]Kainate | >200 (21.5 ± 5.9) | [3H]SR95531 | 83 (68.0 ± 6.9) |
[3H]AMPA | >200 (21.2 ± 9.4) | [3H]rauwolscine | >200 (−2.4 ± 15.0) |
Percentage of displacement obtained in the presence of 200 μM DCUKA is given in parentheses.