Compounds | CB1 | CB1/2(TMIII) | ||
---|---|---|---|---|
EC50 | Maximum Inhibition | EC50 | Maximum Inhibition | |
nM | % | nM | % | |
CP 55,940 | 5.5 ± 2.9 | 72 | 15.8 ± 6.8 | 78 |
WIN 55,212-2 | 38.9 ± 8.2 | 68 | 7.0 ± 0.6 | 97 |
JWH 018 | 14.7 ± 3.9 | 79 | 4.7 ± 0.8 | 70 |
Results are presented as mean ± S.E. of EC50 values from at least two experiments performed in duplicate.