Enzyme | Ki |
---|---|
nM | |
Chymotrypsin | 0.26 |
Elastase | 0.34 |
Tryptase | 0.58 |
Cathepsin G | 11.0 |
Trypsin | 23.6 |
Kallikrein (tissue) | No inhibition at 83 μM |
Thrombin | No inhibition at 83 μM |
Factor Xa | No inhibition at 100 μM |
Kallikrein (plasma) | No inhibition at 100 μM |
Plasmin | No inhibition at 100 μM |