Chemical structures, calculated log Poct, transepithelial permeability coefficient, cell partitioning, and mass balance of pyrrolopyrimidine analogs assayed using MDCK cell monolayers
↵1-a Calculated log Poct/water.
↵1-b Apparent permeability coefficient × 10−6(cm/s).
↵1-c Percent of donor mass equilibrating with the cell monolayer.
1-150 Some metabolism detected.