Organic Cation | Km | Vmax | |
---|---|---|---|
μM | nmol/mg/min | ||
Amiloride | 7.5 | 5 | Wright and Wunz (1989) |
Choline | 10,000 | 38 | Wright et al. (1992) |
Cimetidine | 4.6 | 0.4 | Gisclon et al. (1987) |
Guanidine | 280 | 1.7 | Miyamoto et al. (1989) |
3400 | 11.2 | ||
MPP+ | 7.8 | 3.3 | Lazaruk and Wright (1990) |
NMN | 630 | 5.1 | Wright (1985) |
2620 | 7.0 | Ott et al. (1991) | |
Procainamide | 540 | 2.8 | McKinney and Kunneman (1985) |
Quinidine | 2.52-a | Ott et al. (1991) | |
Quinine | 2.42-a | Ott et al. (1991) | |
TEA | 490 | 2.7 | Miyamoto et al. (1989) |
↵2-a Apparent Kt.