Table 1

Displacement of [3H]CP55,940 and [3H]SR141716A

Compound[3H]CP55,940Compound[3H]SR141716A
KiS.E.M.nKiS.E.M.n
nM nM
CP-55,9400.540.039SR141716A1.180.109
4′-I-SR141716A2.420.0734′-I-SR141716A1.270.093
WIN55212-22.480.2934′-Br-SR141716A2.040.516
4′-Br-SR141716A2.961.126CP-55,94020.74.836
SR141716A6.181.205WIN55212-221.86.064
Anandamide29.77.4944′,6-I2-SR141716A62.69.794
Δ9-THC37.02.9854′-H-SR141716A71.510.03
4′-H-SR141716A80.916.44Anandamide10310.83
4′,6-I2-SR141716A12619.456-I-SR141716A10812.03
6-I-SR141716A16628.244′,3-I2-SR141716A11356.64
4′,3-I2-SR141716A19836.04Δ9-THC11918.93
Cannabinol24718.143-I-SR141716A19732.93
3-I-SR141716A28232.93Cannabinol74368.13
Cannabidiol22834534Cannabidiol12581473