Formulation | IC50 | S.E. | Hill coefficient | S.E. | n | |
---|---|---|---|---|---|---|
nM | ||||||
MRZ 2/499 | Acid | 2991.1 | 280.1 | 1.11 | 0.05 | 4 |
MRZ 2/577 | Choline salt | 3857.6 | 247.2 | 1.04 | 0.04 | 4 |
MRZ 2/502 | Acid | 90.9 | 0.85 | 1 | ||
MRZ 2/576 | Choline salt | 100.7 | 14.2 | 0.93 | 0.02 | 4 |
MRZ 2/514 | Acid | 106.3 | 0.91 | 1 | ||
MRZ 2/570 | Choline salt | 104.0 | 16.1 | 0.95 | 0.03 | 4 |
MRZ 2/516 | Acid | 626.2 | 0.89 | 1 | ||
MRZ 2/571 | Choline salt | 778.8 | 123.5 | 0.98 | 0.02 | 6 |
L-701,324 | 3.88 | 0.23 | 1.14 | 0.02 | 4 | |
L-689,560 | 6.74 | 0.38 | 1.13 | 0.07 | 4 | |
DCKA1-b | 80.1 | 17.5 | 0.90 | 0.04 | 7 | |
5,7-DiCl-thio-KA | 116.8 | 4.9 | 1.08 | 0.20 | 4 | |
7-Cl-thio-KA | 146.2 | 11.4 | 1.05 | 0.05 | 4 | |
Kynurenic acid | 7970.0 | 1.00 | 1 | |||
Glycine | 304.0 | 89.4 | 0.84 | 0.01 | 5 | |
d-Serine | 354.3 | 172.3 | 0.88 | 0.01 | 4 | |
l-Serine | 25350.0 | 2757.7 | 0.98 | 0.03 | 3 | |
ACPC1-c | 312.5 | 22.2 | 0.78 | 0.06 | 4 | |
(+R)-HA-966 | 1810.0 | 0.83 | 1 |