Receptor | Ligand | Ki(nM) |
---|---|---|
Muscarinic | [3H]Oxotremorine-M | >10,000 |
Adenosine | [3H]NECA | >10,000 |
Alpha-1 | [3H]Prazosin | >10,000 |
Alpha-2 | [3H]RX 781094 | >10,000 |
Beta-1 | [125I]iodo-pindolol | >10,000 |
Beta-2 | [125I]iodo-pindolol | >10,000 |
Dopamine | [3H]Spiperone | >10,000 |
Glutamate | [3H]Glutamate | >10,000 |
Quisqualate | [3H]AMPA | >10,000 |
Kainate | [3H]Kainic acid | >10,000 |
MK-801 | [3H]MK-801 | >10,000 |
NMDA | [3H]CGS 19755 | >10,000 |
PCP | [3H]TCP | >10,000 |
Glycine, nonstrychnine | [3H]Glycine | >10,000 |
Sigma | [3H]Di(2-tolyl)guanidine | >10,000 |
Glycine, strychnine | [3H]Strychnine | >10,000 |
GABAA | [3H]GABA | >10,000 |
GABAB | [3H]GABA (+50 mM isoguvacine to block GABAA) | >10,000 |
Benzodiazepine (peripheral) | [3H]PK11195 | >10,000 |
Benzodiazepine (central) | [3H]Flunitrazepam | >10,000 |
Serotonin | [3H]dLSD | >10,000 |
Serotonin3 | [3H]GR65630 | >10,000 |
Opioid | [3H]Naloxone | >10,000 |
Bradykinin | [3H]Bradykinin | >10,000 |
Endothelin A | [125I]Endothelin | >10,000 |
Endothelin B | [125I]Endothelin | >10,000 |
Neurokinin 1 (Substance P) | [4,5-3H-Leu]Substance P | >10,000 |
Neuropeptide Y | [125I]Neuropeptide Y | >10,000 |
Neurotensin | [3H]Neurotensin | >10,000 |
VIP | [125I]VIP | >10,000 |
Calcium channel (Type N) | [125I]ω-Conotoxin | >10,000 |
Calcium channel (Type T,L) | [3H]Nitrendipine | >10,000 |
Chloride channel, TBOB | [3H]TBOB | >10,000 |
Potassium channel, apamin | [125I]Apamin | >10,000 |
Potassium channel (ATP modulatory) | [3H]Glibenclamide | >10,000 |
Potassium (voltage dependent) | [125I]Charybdotoxin | >10,000 |
Norepinephrine uptake | [3H]Desmethylimipramine | >10,000 |
Serotonin uptake | [3H]Citalopram | >10,000 |
GABA uptake | [3H]GABA | >10,000 |
Choline uptake | [3H]Choline chloride | >10,000 |
Dopamine, cocaine site | [3H]WIN 35,428 | >10,000 |
Protein kinase C | [3H]Phorbol ester dibutyrate | >10,000 |
Acetylcholinesterase | >10,000 | |
Monoamine oxidase A | [14C]5-HT | >10,000 |
Monoamine oxidase B | [14C]PEA | >10,000 |
Abbreviations: NMDA, N-methyl-d-aspartate; PCP, phencyclidine; GABA, γ-aminobutyric acid; 5-HT, 5-hydroxytryptamine; AMPA, (±)-α-amino-3-hydroxy-5-methylisoxazole-4-propionic acid; NECA, 1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-β-l-ribofuranuronamide; PEA, phenylethylamine; TBOB, 1-phenyl-4-t-butyl-2,6,7-trioxabicyclo(2,2,2)octane.