Daunomycin Vehicle | Vehicle1-a | AUC060 min | AUC0∞ | ||
---|---|---|---|---|---|
Lipo | PEG | IgG | (%ID ∗ min/ml)1-b | (%ID ∗ min/ml)1-b | |
Free drug | − | − | − | 5.5 ± 0.9 | 6.6 ± 0.9 |
Liposomes | + | − | − | 34.9 ± 10.9 | 42.9 ± 14.3 |
PEG-liposomes | + | + | − | 557.1 ± 46.7 | 1880.9 ± 26.0 |
IgG2a | + | + | + | 347.3 ± 27.9 | 795.8 ± 134.9 |
OX2629 | + | + | + | 196.4 ± 19.3 | 316.7 ± 34.9 |
OX26197 | + | + | + | 196.2 ± 5.1 | 401.4 ± 21.7 |
OX26197 + 1 mg OX26 | + | + | + | 460.5 ± 27.8 | 1228.5 ± 132.7 |