Table 4

Ki (nM) determinations with [3H]NGD 94-1 at recombinant human D4.2, D4.4 and D4.7receptor variants expressed in CHO cells4-a

CompoundD4.2D4.4D4.7
NGD 94-14.22.22.1
Octoclothepin0.80.50.9
Haloperidol4-b 10.02.97.1
Clozapine4-b 83.036.061.0
  • 4-a K d (nM) values for human D4.2, D4.4 and D4.7 receptor variants were 1.4, 1.7 and 1.1 nM, respectively.

  • 4-b Data reported in Hill et al. (1996).