Isolated Hepatocytes | Liver Perfusion (MID) | In vivo (LUR, DB model)6-a | In vivo (LUR, DP model)6-a | |||||
---|---|---|---|---|---|---|---|---|
PSu,inf6-b | PSu,inf6-c | fp · PSu,inf | PSu,inf | fb · PSu,inf | PSu,inf | fb · PSu,inf | PSu,inf | |
μl/min/106 | ml/min/g | ml/min/g | ml/min/g | ml/min/g | ml/min/g | ml/min/g | ml/min/g | |
Glucuronide | 41.0 ± 9.0 | 4.92 ± 1.08 | 1.20 ± 0.17 | 4.19 ± 0.59 | 1.67 ± 0.32 | 2.64 ± 0.50 | 1.82 ± 0.36 | 2.85 ± 0.56 |
Sulfate | 320 ± 1 | 38.4 ± 0.1 | 0.74 ± 0.14 | 11.5 ± 2.1 | 1.53 ± 0.08 | 15.6 ± 0.8 | 1.63 ± 0.08 | 16.7 ± 0.9 |