Drug | Ki (nM) | ||||
---|---|---|---|---|---|
D2 Receptor Family | D1Receptor Family | ||||
D2 | D3 | D4 | D1 | D5 | |
Amisulpride | 2.8 | 3.2 | >1000 | >1000 | >1000 |
Haloperidol | 0.60 | 2.3 | 3.8 | 271-a | 481-a |
Clozapine | 80 | 230 | 89 | 1411-a | 2501-a |
Studies of radioligand binding to human dopamine receptor subtypes transfected into CHO (D2 receptor family) or Sf9 (D1 receptor family) cells were performed as described in “Materials and Methods”. Data represent the mean of at least two independent experiments performed in duplicate.
↵1-a , Data taken from Sunahara et al. (1991).