Agonist | Estimated Parameters | ||||
---|---|---|---|---|---|
Log Ka | Log RIia | Log RAia | Log Kobs | Relative τb | |
Oxotremorine-M | N.D. | N.D. | 2.01 | 5.46 | 1.00 |
Oxotremorine | 5.96 | 0.74 | 1.77 | 6.02 | 0.16 |
Carbachol | 5.17 | −0.05 | 1.43 | 5.31 | 0.37 |
Arecoline | 5.44 | 0.22 | 1.37 | 5.51 | 0.20 |
S-Aceclidine | 5.35 | 0.13 | 1.13 | 5.40 | 0.15 |
Pilocarpine | 5.54 | 0.32 | 0.75 | 5.55 | 0.044 |
R-Aceclidine | 5.01 | −0.21 | 0.38 | 5.03 | 0.063 |
Bethanechol | 4.09 | −1.13 | 0.27 | 4.21 | 0.32 |
McN-A-343 | 5.22 | 0.00 | 0.00 | 5.23 | 0.017 |