Metabolite | CBR Polymorphism | Uptake μM | Retention μM |
---|---|---|---|
DOXOL | − | n.d. | n.d. |
+ | n.d. | n.d. | |
EPIOL | − | n.d. | n.d. |
+ | n.d | n.d. | |
DNROL | − | 0.110 ± 0.032 | 0.048 ± 0.010 |
+ | 0.221 ± 0.065 | 0.096 ± 0.018 | |
IDAOL | |||
Day 1 | − | n.a. | 0.015 ± 0.004 |
+ | n.a. | 0.029 ± 0.003 | |
Day 2 | − | n.a. | 0.023 ± 0.004 |
+ | n.a. | 0.035 ± 0.011 | |
Day 3 | − | n.a. | 0.041 ± 0.013 |
+ | n.a. | 0.081 ± 0.030 | |
Cumulative | − | n.a. | 0.078 ± 0.010 |
+ | n.a. | 0.160 ± 0.019 |
n.d., Not detectable.