TABLE 2
Mouse pharmacokinetic results for VU0477573
Dose
Time
Unbound Plasma
Unbound Brain
mg/kg
1
h
nM
nM
1
0.25
36.4
27.7
0.75
16.4
20.9
3
0.25
69.7
53.7
0.75
82.0
43.7
10
0.25
302
239
0.75
335
164
30
0.25
1009
670
0.75
783
569