Compound | IC50 ± S.E.M. |
---|---|
nM | |
(+)-Butaclamol | 160 ± 31 |
Amitriptyline | 7.2 ± 1.2 |
Amperozide | 570 ± 110 |
Aripiprazole | 6500 ± 770 |
Asenapine | 0.30 ± 0.06 |
Benztropine | 340 ± 41 |
Chlorpromazine | 17 ± 0.88 |
Chlorprothixene | 1.2 ± 0.39 |
Cis-(Z)-flupenthixol | 0.35 ± 0.07 |
Clozapine | 14 ± 2.9 |
Cyproheptadine | 6.5 ± 1.9 |
Diphenhydramine | 7500 ± 2800 |
Haloperidol | 4300 ± 1000 |
Ketanserin | 3200 ± 360 |
Ketotifen | 750 ± 180 |
Loratadine | 18,000 ± 1800 |
Loxapine | 5.9 ± 1.4 |
LY-310,762 | 3000 ± 820 |
Methiothepin | 0.25 ± 0.05 |
Mianserin | 130 ± 24 |
Olanzapine | 11 ± 2.2 |
Pirenperone | 680 ± 98 |
R59-022 | 53 ± 13 |
Risperidone | 150 ± 41 |
Ritanserin | 500 ± 110 |