Compound | IC50 ± S.E.M. | Relative Fold Selectivity (AaDOP2/hD1) |
---|---|---|
nM | ||
Amitriptyline | 1100 ± 110 | 170 |
Amperozide | 13000 ± 680 | 23 |
Asenapine | 150 ± 11 | 500 |
Chlorpromazine | 750 ± 80 | 44 |
Chlorprothixene | 49 ± 8.5 | 41 |
Cis-(Z)-flupenthixol | 19 ± 1.7 | 54 |
Cyproheptadine | 1400 ± 160 | 220 |
Doxepin | 2500 ± 240 | 130 |
Loxapine | 300 ± 31 | 51 |
Methiothepin | 83 ± 9.0 | 330 |
SCH-23390 | 1.2 ± 0.20 | 0.0009 |