CEREP BioPrint In Vitro Pharmacology Profile for all hits >15% effect at 10 μM
| Target | % Inhibition | CEREP Catalog Reference |
|---|---|---|
| CCK2 (human) | 35 | 824-2h |
| Melatonin 2 (hamster) | 32 | 892-2 |
| Na+ channel (site 2) (rat) | 32 | 862-a |
| Serotonin 5-HT2b (human) | 26 | 808-2bah |
| μ-Opioid (human) | 25 | 843-h |
| Choline transporter 1 (human) | 22 | 806-Uh |
| Adrenergic α2b (human) | 21 | 802-1bAh |
| Cyclooxygenase 2 (human) | 21 | 777-2hr |
| Muscarinic M3 (human) | 21 | 806-3h |
| κ-Opioid (rat) | 20 | 842-r |
| Neurokinin 1 (human) | 18 | 826-1h |
CCK2, cholecystokinin receptor 2.