Assay | Species | IC50 | S.E.M. | n |
---|---|---|---|---|
nM | ||||
TRPM8 WS-12 activation | Human | 181 | 7.21 | 25 |
TRPM8 cold activation | Human | 480 | 42.76 | 13 |
TRPM8 voltage activation at room temperature | Human | 103 | 29.4 | 3–4 |
TRPM8 voltage activation at room temperature | Guinea pig | 109 | 38.8 | 3 |
TRPM8 voltage activation at 12°C | Human | 13.8 | 2.2 | 3–4 |
TRPM8 WS-12 activation (transients) | Human | 29.6 | 14.8 | 3 |
TRPM8 WS-12 activation (transients) | Rat | 19.3 | 7.1 | 3 |
TRPM8 WS-12 activation (transients) | Guinea pig | 43.5 | n/a | 2 |
n/a, not applicable.