Ligand | pEC50 (Mean ± S.E.M.) in Cells Expressing: | |||
---|---|---|---|---|
DOR333-Gqi4 + DOR | MOR354-Gqi4 + DOR | DOR333-Gqi4 + MOR | MOR354-Gqi4 + MOR | |
Deltorphin II | 7.8 ± 0.1 | 7.3 ± 0.3 | 7.9 ± 0.1 | <5 |
SNC80 | 7.7 ± 0.2 | 7.2 ± 0.2 | 7.0 ± 0.3 | <5 |
ARM1000390 | 6.9 ± 0.2 | 6.5 ± 0.1 | 6.4 ± 0.1 | <5 |
ADL5859 | 6.7 ± 0.1 | 5.9 ± 0.3 | 5.8 ± 0.2* | <5 |
↵* P < 0.05 vs. DOR333-Gqi4 + WT DOR.