TABLE 2
Serum stability of AngIV analogs
Values are the mean ± S.D. (
N
= 3).
Compound
Half-Life
min
Nle
1
-AngIV
1.42 ± 0.26
N
-Acetyl-Nle-Tyr-Ile-His
115 ± 7.6
d
-Nle-Tyr-Ile
225 ± 23.7
GABA-Tyr-Ile
946 ± 234
Nle-Tyr-Ile-His-NH
2
23.0 ± 3.1
Dihexa
335.5 ± 9.5