TABLE 1

Ki values (μM) for OC000459 for DP2 binding compared with other prostanoid receptors

Ki or IC50
Human DP2Rat DP2DP1TPEP1EP2EP3EP4FPIP
Mean0.0130.003>10>10>10>10>10>10>10>10
S.E.M.0.0020.001
n13574355433
  • FP, prostaglandin F receptor; IP, prostacyclin receptor.