TABLE 3

Plasma concentrations of GSK1521498 after oral administration

GSK1521498 was administered by oral gavage at the indicated doses and plasma concentration was determined over a 24-h period.

TimePlasma Concentration
1 mg/kga10 mg/kga
MeanS.D.MeanS.D.
ng/ml
0.25 h583938761
0.5 h110571120240
1 h19897169080
2 h271582060410
4 h305231750170
8 h172221110180
24 h156668
  • a Single administered dose.