TABLE 2
Affinity of GSK1521498 and naltrexone for human and rat MOR, KOR, and DOR
GSK1521498
Naltrexone
fp
K
i
SD
n
fp
K
i
SD
n
Human
μ
8.82
0.09
17
8.33
0.10
4
δ
7.52
0.24
14
7.38
0.14
4
κ
7.69
0.17
14
7.70
0.14
4
Rat
μ
9.14
0.22
12
8.83
0.17
4
δ
7.32
0.24
8
7.45
0.26
4
κ
7.42
0.17
10
7.55
0.21
4