TABLE 1
Best fit values for
Fig. 2
ACh and S 24795 on α7
ACh and Cytisine on (α4)
3
(β2)
2
R
max
n
EC
50
In
max
IC
50
R
max
n
EC
50
In
max
IC
50
μ
M
mM
μ
M
μ
M
Activation
ACh
1.0
1.45
37
1.0
1.5
148
S 24795
0.20
0.85
14
Cytisine
0.35
0.61
88
Inhibition
0.26
1.0
1
1.7
0.7
32